Bioactive Phenolic and Isocoumarin Glycosides from the Stems of Homalium paniculiflorum.

نویسندگان

  • Shou-Yuan Wu
  • Yan-Hui Fu
  • Qi Zhou
  • Meng Bai
  • Guang-Ying Chen
  • Si-Yu Zhao
  • Chang-Ri Han
  • Xiao-Ping Song
چکیده

Two new phenolic glycosides (1 and 2) and two new isocoumarin glycosides (3 and 4), along with 14 known compounds (5-18), were isolated from the stems of Homalium paniculiflorum. Their structures were established on the basis of extensive spectroscopic analyses and chemical methods. All new compounds were evaluated for their anti-inflammatory activities via examining the inhibitory activity on nitric oxide (NO) production induced by lipopolysaccharide (LPS) in mouse macrophage RAW 264.7 cells in vitro. Compounds 1 and 4 exhibited inhibitory activities with IC50 values of 30.23 ± 1.23 μM and 19.36 ± 0.19 μM, respectively.

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عنوان ژورنال:
  • Molecules

دوره 23 2  شماره 

صفحات  -

تاریخ انتشار 2018